Enasidenib

About

Therapy type: Targeted therapy

Therapy strategy: IDH2 inhibition

Mappings

NCI Thesaurus: Enasidenib (ncit:C111573)

Therapeutic response

Precision oncology relationships for therapeutic response involving this therapy.

Type Biomarker(s) Cancer type Therapy(ies)
Sensitivity (+) IDH2 p.R140Q Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R140L Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R140G Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R140W Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R172K Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R172M Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R172G Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R172S Acute Myeloid Leukemia Enasidenib
Sensitivity (+) IDH2 p.R172W Acute Myeloid Leukemia Enasidenib